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Cholesterol occupies the lipid translocation pathway to block phospholipid scrambling by a G protein-coupled receptor
Affiliation:1. Department of Physiology and Biophysics, Weill Cornell Medicine, 1300 York Avenue, Room LC-501C, New York, NY 10065, USA;2. Istituto di Scienze e Tecnologie Chimiche SCITEC, CNR, Via Mario Bianco 9, 20131 Milano, Italy;3. Roivant Sciences, New York, NY 10036, USA;4. Department of Biochemistry, Weill Cornell Medicine, New York, NY 10065, USA;5. Institute for Computational Biomedicine, Weill Cornell Medicine, New York, NY 10065, USA
Abstract:
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  • Keywords:cholesterol  GPCR  Markov State Model  molecular dynamics simulations  rhodopsin  scramblase
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