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Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors
Authors:Wenchao Lu  Huan Xiong  Yu Chen  Chen Wang  Hao Zhang  Pan Xu  Jie Han  Senhao Xiao  Hong Ding  Zhifeng Chen  Tian Lu  Jun Wang  Yuanyuan Zhang  Liyan Yue  Yu-Chih Liu  Chenhua Zhang  Yaxi Yang  Hualiang Jiang  Cheng Luo
Institution:1. State Key Laboratory of Drug Research, CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China;2. Department of Medicinal Chemistry, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China;3. University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing 100049, China;4. Shanghai ChemPartner Co., LTD., Zhangjiang Hi-Tech Park, Shanghai 201203, China;5. Department of Chemistry, College of Sciences, Shanghai University, 99 Shangda Road, Shanghai 200444, China;6. Department of Pharmacy, Guiyang University of Traditional Chinese Medicine, South Dong Qing Road, Guizhou 550025, China;7. Jiangsu Key Laboratory for High Technology Research of TCM Formulae, Nanjing University of Chinese Medicine, 138 Xianlin Road, Nanjing 210023, China;8. School of Life Science and Technology, ShanghaiTech University, 100 Haike Road, Shanghai 201210, China;9. Open Studio for Druggability Research of Marine Natural Products, Pilot National Laboratory for Marine Science and Technology (Qingdao), 1 Wenhai Road, Aoshanwei, Jimo, Qingdao 266237, China
Abstract:
Keywords:Drug discovery  Epigenetics  Histone acetyltransferase  P300/CBP
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