Novel non-peptide ligands for the somatostatin sst3 receptor |
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Authors: | Moinet C Contour-Galcéra M O Poitout L Morgan B Gordon T Rouber P Thurieau C |
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Institution: | Institut Henri Beaufour, Les Ulis, France. christophe.moinet@beaufour-ipsen.com |
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Abstract: | A series of imidazole derivatives has been prepared using high throughput parallel synthesis. Several compounds showed high affinity (Ki in 10(-6)-10(-8) M range) and selectivity at recombinant human somatostatin receptor subtype 3 (hsst3). |
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