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7-Pyrrolidinyl- and 7-piperidinyl-5-aryl-pyrrolo[2,3-d]pyrimidines--potent inhibitors of the tyrosine kinase c-Src
Authors:Altmann E  Missbach M  Green J  Susa M  Wagenknecht H A  Widler L
Institution:Novartis Pharma Research, Arthritis and Bone Metabolism Therapeutic Area, Basel, Switzerland. eva.altmann@pharma.novartis.com
Abstract:7-Heterocyclyl-5-aryl-pyrrolo2,3-d]pyrimidines represent a new class of highly potent and selective inhibitors of the tyrosine kinase pp60(c-Src).
Keywords:
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