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Delineating the conformational landscape of the adenosine A2A receptor during G protein coupling
Authors:Shuya Kate Huang  Aditya Pandey  Duy Phuoc Tran  Nicolas L. Villanueva  Akio Kitao  Roger K. Sunahara  Adnan Sljoka  R. Scott Prosser
Affiliation:1. Department of Chemistry, University of Toronto, UTM, 3359 Mississauga Road North, Mississauga, Ontario L5L 1C6, Canada;2. Department of Biochemistry, University of Toronto, 1 King’s College Circle, Toronto, Ontario M5S 1A8, Canada;3. School of Life Science and Technology, Tokyo Institute of Technology, 2-12-1 Ookayama, Meguro-ku, Tokyo 152-8550, Japan;4. Department of Pharmacology, University of California San Diego School of Medicine, 9500 Gilman Drive, La Jolla, CA 92093, USA;5. RIKEN Center for Advanced Intelligence Project, RIKEN, 1-4-1 Nihombashi, Chuo-ku, Tokyo 103-0027, Japan
Abstract:
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  • Keywords:GPCR  G protein  allostery  precoupling  partial agonism  rigidity transmission allostery
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