aDepartament de Quı´mica Inorgànica i Orgànica, Universitat Jaume I, 12071 Castelló, Spain;bSandler Center for Basic Research in Parasitic Diseases, Box 2550, University of California, San Francisco, San Francisco, CA 94143-2550, USA
Abstract:
The dipeptidyl epoxyesters 3 and 4 are potent, irreversible inhibitors of cruzain and rhodesain.