引用本文: | Frohn M,Cee VJ,Lanman BA,Pickrell AJ,Golden J,Rivenzon-Segal D,Middleton S,Fiorino M,Xu H,Schrag M,Xu Y,McElvain M,Muller K,Siu J,Bürli R.Novel 5- and 6-subtituted benzothiazoles with improved physicochemical properties: potent S1P₁ agonists with in vivo lymphocyte-depleting activity[J].Bioorganic & Medicinal Chemistry Letters,2012,22(1):628-633. |