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Optimization and biological evaluation of thiazole-bis-amide inverse agonists of RORγt
Institution:1. Phenex Pharmaceuticals AG, Waldhofer Strasse 104, 69123 Heidelberg, Germany;2. Janssen Research and Development, LLC, San Diego, CA 92121, USA;3. Janssen Research and Development, Spring House, PA 19477, USA;1. Genentech, Inc., 1 DNA Way, South San Francisco, CA 94080, USA;2. Argenta, Units 7–9 Spire Green Centre, Flex Meadow, Harlow, Essex CM19 5TR, UK;1. Discovery Product Development and Supply, Janssen Research and Development, 3210 Merryfield Row, San Diego, CA 92121, United States;2. Discovery Product Development and Supply, Janssen Research and Development, Welsh and McKean Roads, Spring House, PA 19477, United States;3. Department of Research, Phenex Pharmaceuticals AG, Heidelberg, Germany;4. Discovery Immunology, Janssen Research and Development, 3210 Merryfield Row, San Diego, CA 92121, United States;1. Reata Pharmaceuticals, Inc., 2801 Gateway Drive, Suite 150, Irving, TX 75063, USA;2. Department of Chemistry, Michigan State University, 578 South Shaw Lane, East Lansing, MI 48824, USA
Abstract:
Keywords:Retinoid-related orphan receptor gamma t  RORc  RORgt  Thiazole  Inverse agonist
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