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UM171 Preserves Epigenetic Marks that Are Reduced in Ex Vivo Culture of Human HSCs via Potentiation of the CLR3-KBTBD4 Complex
Authors:Jalila Chagraoui  Simon Girard  Jean-Francois Spinella  Laura Simon  Eric Bonneil  Nadine Mayotte  Tara MacRae  Jasmin Coulombe-Huntington  Thierry Bertomeu  Celine Moison  Elisa Tomellini  Pierre Thibault  Mike Tyers  Anne Marinier  Guy Sauvageau
Institution:1. Molecular Genetics of Stem Cells Laboratory, Institute for Research in Immunology and Cancer (IRIC), Université de Montréal, Montreal, QC, Canada;2. Departments of Biochemistry and Chemistry, Institute for Research in Immunology and Cancer, Université de Montréal, Montreal, QC, Canada;3. Department of Medicine, Institute for Research in Immunology and Cancer (IRIC), Université de Montréal, Montreal, QC, Canada;4. Faculty of Arts and Science, Université de Montréal, Montreal, QC, Canada;5. Division of Hematology, Maisonneuve-Rosemont Hospital, Montreal, QC, Canada;6. Department of Medicine, Faculty of Medicine, Université de Montréal, Montreal, QC, Canada
Abstract:
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  • Keywords:epigenetic modulation  LSD1/RCOR1 CoREST complex  Cullin3 E3 ligase-mediated proteasomal degradation  Kelch-BTB domain proteinUM171 small molecule  HSC self-renewal
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