Benzo[b]thiophene-2-carboxamides and benzo[b]furan-2-carboxamides are potent antagonists of the human H3-receptor |
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| Authors: | Peschke Bernd Bak Sonja Hohlweg Rolf Nielsen Rita Viuff Dorthe Rimvall Karin |
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| Institution: | Novo Nordisk A/S, Novo Nordisk Park, DK-2760 Maaloev, Denmark. bpes@novonordisk.com |
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| Abstract: | Benzob]thiophene-2-carboxamides and benzob]furan-2-carboxamides have been found to be antagonists on the human histamine-3-receptor, showing a Ki value of as low as 4 nM. |
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