Dihydropyrazolopyrimidine Inhibitors of KV1.5 (IKur) |
| |
Institution: | Bristol-Myers Squibb, Route 206 & Provinceline Road, PO Box 4000, Princeton, NJ 08543-4000, USA |
| |
Abstract: | A series of dihydropyrazolopyrimidine inhibitors of KV1.5 (IKur) have been identified. The synthesis, structure–activity relationships and selectivity against several other ion channels are described. |
| |
Keywords: | |
本文献已被 ScienceDirect 等数据库收录! |
|