The action of dibucaine in vitro on fat cell lipolysis and protein kinase activity. |
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Authors: | S Psychoyos H Chertock |
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Institution: | Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation Ardsley, New York 10502, USA |
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Abstract: | Dibucaine at 0.1 and 0.25 mM markedly inhibited epinephrine-stimulated lipolysis in rat epididymal fat cells but did not inhibit protein kinase activity. At 1.0 mM, dibucaine half-maximally stimulated protein kinase of fat cells under basal conditions but did not stimulate lipolysis. It is concluded that dibucaine inhibits lipolysis by a mechanism not involving inhibition of protein kinase. |
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