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4-Aminoarylguanidine and 4-aminobenzamidine derivatives as potent and selective urokinase-type plasminogen activator inhibitors
Authors:Spencer Jeffrey R  McGee Danny  Allen Darin  Katz Bradley A  Luong Christine  Sendzik Martin  Squires Neil  Mackman Richard L
Affiliation:Celera, 180 Kimball Way, South San Francisco, CA 94080, USA.
Abstract:The structure-based design of potent and selective urokinase-type plasminogen activator (uPA) inhibitors with 4-aminoarylamidine or 4-aminoarylguanidine S1 binding groups, is described.
Keywords:
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