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Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants
Authors:Butini Stefania  Gemma Sandra  Brindisi Margherita  Borrelli Giuseppe  Fiorini Isabella  Samuele Alberta  Karytinos Aristotele  Facchini Marcella  Lossani Andrea  Zanoli Samantha  Campiani Giuseppe  Novellino Ettore  Focher Federico  Maga Giovanni
Institution:a European Research Centre for Drug Discovery and Development (NatSynDrugs), via Aldo Moro, 2-Università di Siena, 53100 Siena, Italy
b Dipartimento Farmaco Chimico Tecnologico, via Aldo Moro, 2 - Università di Siena, 53100 Siena, Italy
c DNA Enzymology and Molecular Virology, Institute of Molecular Genetics IGM-CNR, National Research Council, 27100 Pavia, Italy
d Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, via D. Montesano 49, 80131 Napoli, Italy
Abstract:
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