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3H]-(R)-NPTS,a radioligand for the type 1 glycine transporter |
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| Authors: | Lowe John A Drozda Susan E Fisher Katherine Strick Christine Lebel Lorraine Schmidt Christopher Hiller Donna Zandi Kathleen S |
| Affiliation: | Central Research Division, Pfizer Inc., Groton, CT 06340, USA. john_a_lowe@groton.pfizer.com |
| Abstract: | The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine transporter (GlyT1) is described, as well as preparation of 6 in optically active and tritiated form for use as a radioligand for affinity displacement assay of GlyT1. |
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