Design,synthesis, and biological evaluation of substrate-competitive inhibitors of C-terminal Binding Protein (CtBP) |
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Institution: | 1. Department of Medicinal Chemistry, School of Pharmacy, The Institute for Structural Biology, Drug Discovery, and Development, and the Massey Cancer Center, Virginia Commonwealth University, Richmond, VA 23298, United States;2. Division of Hematology, Oncology, & Palliative Care, Department of Human and Molecular Genetics, and the Massey Cancer Center, Virginia Commonwealth University, Richmond, VA 23298, United States;3. Department of Molecular, Cell, & Cancer Biology, University of Massachusetts Medical School, Worcester, MA 01605, United States;4. Department of Biochemistry & Molecular Pharmacology, University of Massachusetts Medical School, Worcester, MA 01605, United States;1. Department of Respiratory and Critical Care Medicine, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan 610041, China;2. State Key Laboratory of Oral Diseases, West China Hospital of Stomatology, West China School of Stomatology, Sichuan University, No. 14, Section 3, Renminnan Road, Chengdu, Sichuan 610041, China;3. School of Chemical Engineering, Sichuan University, Chengdu, Sichuan 610065, China;1. Université Paris-Saclay, CNRS, BioCIS, 92290, Châtenay-Malabry, France;2. Univ. Bordeaux, CNRS, Bordeaux INP, ISM, UMR5255, 351 cours Libération, F-33405, Bordeaux, France;1. Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia;2. Department of Medical Biology, University of Melbourne, Parkville, VIC 3010, Australia |
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