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Tyrosyl-DNA phosphodiesterase inhibitors: Progress and potential
Affiliation:1. Vorozhtsov Institute of Organic Chemistry, Siberian Division, Russian Academy of Sciences, pr. akademika Lavrent’eva 9, Novosibirsk 630090, Russian Federation;2. Novosibirsk State University, Pirogova Str. 2, Novosibirsk 630090, Russian Federation;3. Novosibirsk Institute of Chemical Biology and Fundamental Medicine, Siberian Division, Russian Academy of Sciences, pr. akademika Lavrent’eva 8, Novosibirsk 630090, Russian Federation;1. Novosibirsk Institute of Chemical Biology and Fundamental Medicine, Siberian Branch of the Russian Academy of Sciences, Novosibirsk 630090, Russian Federation;2. N. N. Vorozhtsov Novosibirsk Institute of Organic Chemistry, Siberian Branch of the Russian Academy of Sciences, Novosibirsk 630090, Russian Federation;3. Novosibirsk State University, Novosibirsk 630090, Russian Federation;4. School of Chemical Sciences, University of Auckland, New Zealand;1. N.N. Vorozhtsov Novosibirsk Institute of Organic Chemistry, Siberian Branch, Russian Academy of Sciences, 9, Akademika Lavrentieva Ave., Novosibirsk 630090, Russian Federation;2. Novosibirsk Institute of Chemical Biology and Fundamental Medicine, Siberian Branch of the Russian Academy of Sciences, 8, Akademika Lavrentieva Ave., Novosibirsk 630090, Russian Federation;3. Novosibirsk State University, 2, Pirogova Str., Novosibirsk 630090, Russian Federation;4. School of Chemical Sciences, University of Auckland, New Zealand;1. Griffith Institute for Drug Discovery, Griffith University, Brisbane QLD 4111, Australia;2. Centre for Drug Research and Development, Vancouver, British Columbia V6T1Z3, Canada;1. Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, Building 37, Room 5068, NIH, Bethesda, MD 20892, USA;2. Laboratory of Molecular Biology, Indian Association for the Cultivation of Science, Jadavpur, Kolkata 700032, India;3. Department of Radiation Genetics, Graduate School of Medicine, Kyoto University, Yoshidakonoe, Sakyo-ku 606-8501, Japan
Abstract:
Keywords:DNA repair  Topoisomerase  Camptothecin  Top1 inhibitors  Top2 inhibitors  Tyrosyl-DNA phosphodiesterase  Tdp1  Tdp2  Tdp1 inhibitors  Tdp2 inhibitors  Indenoisoquinolines
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