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Dynamic Imaging of LDH Inhibition in Tumors Reveals Rapid In Vivo Metabolic Rewiring and Vulnerability to Combination Therapy
Institution:1. Urologic Oncology Branch, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, USA;2. Radiation Biology Branch, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, USA;3. Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD 20850, USA;4. Mitochondrial Medicine Laboratory, Department of Pathology, University of Alabama at Birmingham, Birmingham, AL 35294, USA;5. Department of Cell Biology, University of Geneva, 1211 Geneva 4, Switzerland;6. Developmental Therapeutics Branch, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, USA;7. University of New Mexico Health Sciences Center, Albuquerque, NM 87131, USA;8. Leidos Biomedical, Frederick National Laboratory for Cancer Research, Frederick, MD 24060, USA;9. Ludwig Institute for Cancer Research, New York, NY 10017, USA;10. The Wistar Institute, Philadelphia, PA 19104, USA;11. Department of Chemistry, Vanderbilt University, Nashville, TN 37240, USA
Abstract:
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  • Keywords:lactate dehydrogenase  pyruvate metabolism  metabolic flux  cancer  metabolic imaging  hyperpolarized magnetic resonance spectroscopic imaging
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