Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5 |
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Authors: | Contour-Galéra M O Poitout L Moinet C Morgan B Gordon T Roubert P Thurieau C |
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Affiliation: | Institut Henri Beaufour, Les Ulis, France. m-odile.galcera.contour@beaufour-ipsen.com |
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Abstract: | A new preparation of trisubstituted imidazopyrazines and dihydroimidazopyrazines via parallel synthesis using aminoacids and bromoketones resulted in the discovery of non-peptidic sst5 selective agonists. |
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