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Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5
Authors:Contour-Galéra M O  Poitout L  Moinet C  Morgan B  Gordon T  Roubert P  Thurieau C
Affiliation:Institut Henri Beaufour, Les Ulis, France. m-odile.galcera.contour@beaufour-ipsen.com
Abstract:A new preparation of trisubstituted imidazopyrazines and dihydroimidazopyrazines via parallel synthesis using aminoacids and bromoketones resulted in the discovery of non-peptidic sst5 selective agonists.
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