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Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors
Authors:Kim Sora  Jung Jin Kyo  Lee Hyo Seon  Kim Youngjae  Kim Jiyoon  Choi Kihang  Baek Du-Jong  Moon Bongjin  Oh Kwang-Seok  Lee Byung Ho  Shin Kye Jung  Pae Ae Nim  Nam Ghilsoo  Roh Eun Joo  Cho Yong Seo  Choo Hyunah
Institution:a Life/Health Division, Korea Institute of Science and Technology, Seongbuk-gu, Seoul 136-791, Republic of Korea
b Department of Chemistry, Korea University, Seongbuk-gu, Seoul 136-713, Republic of Korea
c Department of Chemistry, College of Natural Sciences, Sangmyung University, Seoul 110-743, Republic of Korea
d Department of Medicinal and Pharmaceutical Chemistry, University of Science and Technology, Daejeon, Republic of Korea
e Department of Chemistry, Sogang University, Seoul, Republic of Korea
f Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea
g College of Pharmacy, The Catholic University of Korea, Seongsim Campus, Bucheon, Gyeonggi-do, Republic of Korea
Abstract:
Keywords:Rheumatoid arthritis  Inflammation  Aminopyrimidine  IKK-2  Kinase inhibitor
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