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Gli1/DNA interaction is a druggable target for Hedgehog‐dependent tumors
Authors:Francesca Ghirga  Federica Aiello  Sara Toscano  Cinzia Ingallina  Mariangela Siler  Danilo Cucchi  Agnese Po  Evelina Miele  Davide D'Amico  Gianluca Canettieri  Enrico De Smaele  Elisabetta Ferretti  Isabella Screpanti  Gloria Uccello Barretta  Maurizio Botta  Bruno Botta  Alberto Gulino  Lucia Di Marcotullio
Affiliation:1. Dipartimento di Chimica e Tecnologie del Farmaco, University La Sapienza, Rome, Italy;2. Department of Chemistry and Industrial Chemistry, University of Pisa, Pisa, Italy;3. Center for Life NanoScience@Sapienza, Istituto Italiano di Tecnologia, Rome, Italy;4. Department of Molecular Medicine, University La Sapienza, Rome, Italy;5. Department of Experimental Medicine, University La Sapienza, Rome, Italy;6. Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy;7. Sbarro Institute for Cancer Research and Molecular Medicine, Temple University, Philadelphia, PA, USA;8. Istituto Pasteur, Fondazione Cenci‐Bolognetti ‐ University La Sapienza, Rome, Italy;9. IRCCS Neuromed, Pozzilli, Italy
Abstract:
Keywords:cancer  Gli inhibitors  Gli1–  DNA interaction  Hedgehog
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